- Active Pharmaceutical Ingredients
- Varenicline tartrate
- Aprepitant, Fosapitant Intermediates
- Fosaprepitant Dimeglumine
- Vildagliptin
- Efinaconazole
- Luliconazole Intermediate
- Gadoterate Meglumine
- Succinyl Alcohol Intermediate
- Mirabillon Intermediate
- Atazanavir Intermediate
- Intermediate
- Varenicline tartrate
- Aprepitant 287930-73-8
- Aprepitant 127852-28-2
- Aprepitant 287930-75-0
- Aprepitant 200000-59-5
- Aprepitant 155742-64-6
- Aprepitant 252742-72-6
- Fosaprepitant Dimeglumine 990-91-0
- Fosaprepitant Dimeglumine 265121-01-5
- Vildagliptin 207557-35-5
- Vildagliptin 702-82-9
- Efinaconazole 144230-50-2
- Efinaconazole 133775-25-4
- Efinaconazole 127000-90-2
- Gadoterate Meglumine
- Mirabegron
- Luliconazole 98873-55-3
- Luliconazole 126534-31-4
- Atazanavir sulfate
- Bortezomib 179324-87-9
- Bortezomib 114457-94-2
- Bortezomib 205393-22-2
- Brinzolamide
- Rivaroxaban Intermediate 446292-08-6
- Rivaroxaban Intermediate 446292-07-5
- Cinacalcet Hydrochloride 1005450-55-4
- Cinacalcet Hydrochloride 585-50-2
- Eletriptan Intermediate
- Indacaterol intermediate 312753-53-0
- Indacaterol intermediate 173140-90-4
- Sitagliptin Intermediate
- Fosanavir Calcium Intermediate
Popular information
福沙匹坦中间体 福沙匹坦二苄酯 265121-01-5
English Name :
CAS# :
产品描述
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福沙匹坦二苄酯
Fosaprepitant dibenzyl ester
CAS 265121-01-5
别 名 |
福沙匹坦中间体 |
CAS # |
265121-01-5 |
分子式 |
C37H34F7N4O6P |
分子量 |
794.65 |
结构式 |
|
产品简介 CAS 265121-01-5 |
福沙匹坦二苄酯,英文名为Fosaprepitant dibenzyl ester,美国化学文摘登记号为cas 265121-01-5。 焦磷酸四苄酯(cas 265121-01-5)是福沙吡坦中间体,福沙吡坦是阿瑞匹坦(aprepitant)口服制剂的前体药物,注射后在体内迅速转化成阿瑞吡坦。福沙匹坦二甲葡胺与阿瑞匹坦属于称作人P物质/神经激肽1(NK-1)选择性高亲和性受体阻断剂,主要通过阻断大脑恶心和呕吐信号新颖的作用机制发挥作用。阿瑞匹坦对5-羟色胺(5-HT3)、多巴胺和糖皮质激素受体极微弱或无亲和性,用于治疗化疗诱导的恶心和呕吐及术后恶心和呕吐。 |
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